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  1. Liver Toxicity Knowledge Base (LTKB)

Drug-Induced Liver Injury Severity and Toxicity (DILIst) Dataset

The largest drug list with DILI classification

The drug-induced liver injury severity and toxicity (DILIst) dataset consists of 1,279 drugs that are divided into two classes according to their potential for causing drug-induced liver injury (DILI). The DILI classification was derived from augmenting the DILIrank dataset with four literature datasets that were found to have ≥ 350 drugs with human DILI classification, to generate the largest drug list with DILI classification.

  • 768 DILI Positive
  • 511 DILI Negative

Please let us know if you download the file by contacting NCTRBioinformaticsSupport@fda.hhs.gov.

Reference

Drug-induced liver injury severity and toxicity (DILIst): binary classification of 1279 drugs by human hepatotoxicity.
Thakkar S., Li T., Liu Z., Wu L., Roberts R., and Tong W.
Drug Discovery Today. 2020, 25(1), 201-208.

Contact Information

Questions or Suggestions: Weida Tong, Ph.D. (Weida.Tong@fda.hhs.gov).


*Classification: 0 = DILI Negative; 1 = DILI Positive

DILIST_ID Compound Name DILIst Classification Routes of Administration
1 mercaptopurine 1 Oral
2 acetaminophen 1 Oral
3 azathioprine 1 Oral
4 chlorpheniramine 0 Oral
5 clofibrate 1 Oral
6 cyclophosphamide 1 Oral
7 dopamine 0 Intravenous
8 estradiol 1 Oral
9 fluoxetine 1 Oral
10 gemfibrozil 1 Oral
11 indomethacin 1 Oral
12 ketoprofen 1 Oral
13 mannitol 0 Intravenous
14 methotrexate 1 Oral
15 phenobarbital 1 Oral
16 phenytoin 1 Oral
17 rifampin 1 Oral
18 tetracycline 1 Oral
19 abacavir 1 Oral
20 aciclovir 1 Oral
21 allopurinol 1 Oral
22 amineptine 1 Oral
23 amiodarone 1 Oral
24 amitriptyline 1 Oral
25 amphotericin b 1 Intravenous
26 ampicillin 1 Oral
27 donepezil 1 Oral
28 aspirin 1 Oral
29 aminohippurate 0 Intravenous
30 bicalutamide 1 Oral
31 bupropion 1 Oral
32 captopril 1 Oral
33 carbamazepine 1 Oral
34 carboplatin 1 Intravenous
35 ceftazidime 1 Intravenous
36 chlorcyclizine 1 Oral
37 chlorzoxazone 1 Oral
38 chlorpromazine 1 Oral
39 cisplatin 1 Intravenous
40 dimercaprol 0 Intramuscular
41 colchicine 0 Oral
42 corticotropin 0 Subcutaneous
43 dactinomycin 1 Subcutaneous
44 dantrolene 1 Oral
45 demeclocycline 0 Oral
46 propoxyphene 1 Oral
47 diclofenac 1 Oral
48 diflunisal 1 Oral
49 diphenhydramine 0 Oral
50 epirubicin 0 Intravenous
51 erythromycin 1 Oral
52 etoposide 1 Oral
53 famotidine 1 Oral
54 felbamate 1 Oral
55 fenofibrate 1 Oral
56 fenoprofen 1 Oral
57 flutamide 1 Oral
58 hydroxyurea 1 Oral
59 imatinib 1 Oral
60 imipramine 1 Oral
61 iproniazid 1 Oral
62 ketoconazole 1 Oral
63 labetalol 1 Oral
64 leflunomide 1 Oral
65 mefenamic acid 1 Oral
66 meloxicam 1 Oral
67 metformin 1 Oral
68 methyldopa 1 Oral
69 nefazodone 1 Oral
70 nitrofurantoin 1 Oral
71 olsalazine 1 Oral
72 paroxetine 1 Oral
73 pentamidine 1 Intravenous
74 perhexiline 1 Oral
75 physostigmine 0 Intravenous
76 pioglitazone 1 Oral
77 propylthiouracil 1 Oral
78 pseudoephedrine 0 Oral
79 ranitidine 1 Oral
80 rifabutin 1 Oral
81 rosiglitazone 1 Oral
82 indocyanine green 0 Intravenous
83 simvastatin 1 Oral
84 spironolactone 1 Oral
85 stavudine 1 Oral
86 streptomycin 0 Intramuscular
87 sulfadiazine 1 Oral
88 sulfasalazine 1 Oral
89 sulindac 1 Oral
90 tamoxifen 1 Oral
91 temozolomide 1 Oral
92 theophylline 0 Oral
93 tizanidine 1 Oral
94 tolcapone 1 Oral
95 valproic acid 1 Oral
96 vancomycin 1 Oral
97 vitamin a 1 Intramuscular
98 zidovudine 1 Oral
99 zolpidem 0 Oral
100 zonisamide 1 Oral
101 pyrazinamide 1 Oral
102 finasteride 1 Oral
103 troglitazone 1 Oral
104 fluvastatin 1 Oral
105 glimepiride 1 Oral
106 venlafaxine 1 Oral
107 amlodipine 1 Oral
108 vinblastine 0 Intravenous
109 ciprofloxacin 1 Oral
110 fluconazole 1 Oral
111 prednisone 1 Oral
112 lorazepam 0 Oral
113 itraconazole 1 Oral
114 raloxifene 0 Oral
115 mifepristone 0 Oral
116 clomipramine 1 Oral
117 pravastatin 1 Oral
118 clarithromycin 1 Oral
119 hydrocortisone 0 Oral
120 progesterone 1 Oral
121 ergocalciferol 0 Oral
122 ibuprofen 1 Oral
123 isoproterenol 0 Intravenous
124 ketorolac 1 Oral
125 promethazine 1 Oral
126 omeprazole 1 Oral
127 carvedilol 1 Oral
128 cytarabine 1 Intravenous
129 pergolide 0 Oral
130 nisoldipine 0 Oral
131 citalopram 1 Oral
132 methyltestosterone 1 Oral
133 testosterone 1 Oral
134 praziquantel 0 Oral
135 ticlopidine 1 Oral
136 diazepam 0 Oral
137 clomiphene 1 Oral
138 isotretinoin 1 Oral
139 oxymetholone 1 Oral
140 etodolac 1 Oral
141 glipizide 1 Oral
142 pemoline 1 Oral
143 clotrimazole 1 Oral
144 celecoxib 1 Oral
145 amoxapine 0 Oral
146 iothalamate sodium 0 Intravenous
147 atorvastatin 1 Oral
148 olanzapine 1 Oral
149 nevirapine 1 Oral
150 primidone 0 Oral
151 vinorelbine 0 Intravenous
152 anastrozole 1 Oral
153 rabeprazole 1 Oral
154 azithromycin 1 Oral
155 tolazamide 1 Oral
156 quetiapine 1 Oral
157 famciclovir 0 Oral
158 atenolol 1 Oral
159 benzbromarone 1 Oral
160 bromocriptine 1 Oral
161 busulfan 1 Oral
162 chlorambucil 1 Oral
163 clozapine 1 Oral
164 dacarbazine 1 Intravenous
165 dapsone 1 Oral
166 digoxin 0 Oral
167 disulfiram 1 Oral
168 enalapril 1 Oral
169 furosemide 0 Oral
170 gabapentin 1 Oral
171 glibenclamide 1 Oral
172 isoniazid 1 Oral
173 lansoprazole 1 Oral
174 mebendazole 1 Oral
175 metoprolol 1 Oral
176 naltrexone 0 Oral
177 niacin 1 Oral
178 nifedipine 1 Oral
179 nimesulide 1 Oral
180 nizatidine 1 Oral
181 dextrose 0 Intravenous
182 cholestyramine 0 Oral
183 sodium lactate 0 Intravenous
184 verapamil 1 Oral
185 doxorubicin 1 Intravenous
186 clorazepate 0 Oral
187 protirelin 0 Intravenous
188 sincalide 0 Intravenous
189 secretin 0 Intravenous
190 sucralfate 0 Oral
191 cupric chloride 0 Intravenous
192 trientine hydrochloride 0 Oral
193 chlorpropamide 1 Oral
194 cyclosporine 1 Oral
195 decitabine 0 Intravenous
196 deferoxamine 1 Intravenous
197 doxycycline 1 Oral
198 exemestane 1 Oral
199 felodipine 1 Oral
200 fludrocortisone 0 Oral
201 fluphenazine 0 Oral
202 gefitinib 1 Oral
203 haloperidol 1 Oral
204 mesalazine 1 Oral
205 minocycline 1 Oral
206 ioversol 0 Intravenous
207 oxaprozin 1 Oral
208 paclitaxel 1 Intravenous
209 phentolamine 0 Intravenous
210 prazosin 0 Oral
211 prochlorperazine 1 Oral
212 corticorelin ovine triflutate 0 Intravenous
213 sodium thiosulfate 0 Intravenous
214 sirolimus 1 Oral
215 tacrolimus 1 Oral
216 thalidomide 1 Oral
217 thioridazine 1 Oral
218 thioguanine 1 Oral
219 tolbutamide 0 Oral
220 topiramate 1 Oral
221 trifluoperazine 0 Oral
222 triptorelin pamoate 1 Intramuscular
223 alatrofloxacin mesylate 1 Oral
224 vorinostat 0 Oral
225 nesiritide 0 Intravenous
226 ganirelix acetate 0 Subcutaneous
227 gemtuzumab ozogamicin 1 Intravenous
228 methylprednisolone 1 Oral
229 gamma hydroxybutyric acid 0 Oral
230 tegaserod 0 Oral
231 penicillamine 1 Oral
232 pramlintide 0 Subcutaneous
233 lanthanum carbonate 0 Oral
234 acetazolamide 1 Oral
235 albendazole 1 Oral
236 alprazolam 1 Oral
237 altretamine 0 Oral
238 amantadine 0 Oral
239 4-aminosalicylic acid 1 Oral
240 amoxicillin 1 Oral
241 atropine 0 Intravenous
242 benoxaprofen 1 Oral
243 emtricitabine 0 Oral
244 trospium 0 Oral
245 bromfenac 1 Oral
246 gadofosveset trisodium 0 Intravenous
247 clonazepam 1 Oral
248 exenatide 0 Subcutaneous
249 entecavir 0 Oral
250 danazol 1 Oral
251 daunorubicin 0 Intravenous
252 dimenhydrinate 0 Intravenous
253 doxapram 0 Intravenous
254 febuxostat 1 Oral
255 granisetron 0 Oral
256 griseofulvin 1 Oral
257 hydralazine 1 Oral
258 ibufenac 1 Oral
259 ifosfamide 1 Intravenous
260 deferasirox 1 Oral
261 sunitinib 1 Oral
262 ivermectin 1 Oral
263 lamivudine 1 Oral
264 methylnaltrexone bromide 0 Subcutaneous
265 letrozole 1 Oral
266 desvenlafaxine 1 Oral
267 lomefloxacin 0 Oral
268 lomustine 1 Oral
269 lovastatin 1 Oral
270 telbivudine 0 Oral
271 methimazole 1 Oral
272 methocarbamol 0 Oral
273 metronidazole 1 Oral
274 minoxidil 0 Oral
275 mitomycin 1 Intravenous
276 modafinil 1 Oral
277 fesoterodine 0 Oral
278 naloxone 0 Intravenous
279 naproxen 1 Oral
280 nateglinide 0 Oral
281 neomycin 0 Oral
282 levocetirizine dihydrochloride 1 Oral
283 nystatin 0 Oral
284 oxytetracycline 0 Oral
285 pantoprazole 1 Oral
286 prednisolone 1 Oral
287 primaquine 0 Oral
288 procarbazine 1 Oral
289 ambrisentan 0 Oral
290 secobarbital 0 Oral
291 sertraline 1 Oral
292 sotalol 0 Oral
293 sulfathiazole 1 Oral
294 terbinafine 1 Oral
295 thiabendazole 1 Oral
296 ticrynafen 1 Oral
297 tinidazole 1 Oral
298 maraviroc 1 Oral
299 raltegravir 1 Oral
300 clevidipine 0 Intravenous
301 trovafloxacin 1 Oral
302 regadenoson 0 Intravenous
303 warfarin 1 Oral
304 zaleplon 0 Oral
305 zileuton 1 Oral
306 ferumoxytol 0 Intravenous
307 etravirine 1 Oral
308 silodosin 0 Oral
309 fospropofol 1 Intravenous
310 bendamustine 0 Intravenous
311 tolvaptan 1 Oral
312 eltrombopag olamine 1 Oral
313 tapentadol 0 Oral
314 prasugrel hydrochloride 1 Oral
315 saxagliptin 0 Oral
316 romidepsin 0 Intravenous
317 dronedarone 1 Oral
318 pazopanib 1 Oral
319 pancrelipase 0 Oral
320 dexchlorpheniramine 0 Oral
321 ecallantide 0 Subcutaneous
322 divalproex sodium 1 Oral
323 lumiracoxib 1 Oral
324 tasosartan 1 Oral
325 oxyphenisatin 1 Oral
326 tilbroquinol 1 Oral
327 alclofenac 1 Oral
328 aplaviroc  1 Oral
329 clomacran 1 Oral
330 dermatan 1 Intravenous
331 isaxonine 1 Oral
332 pipamazine 1 Oral
333 pralnacasan  1 Oral
334 sulfacarbamide 1 Oral
335 triacetyldiphenolisatin 1 Oral
336 fiduxosin  1 Oral
337 pafuramidine  1 Oral
338 phenoxypropazine 1 Oral
339 histamine diphosphate 0 Subcutaneous
340 aminophylline 0 Oral
341 meperidine 0 Oral
342 methamphetamine 0 Oral
343 methadone 0 Oral
344 hyaluronidase 0 Subcutaneous
345 doxylamine 0 Oral
346 protamine sulfate 0 Intravenous
347 bethanechol 0 Oral
348 cortisone acetate 0 Oral
349 dicyclomine 0 Oral
350 norepinephrine 0 Intravenous
351 dyphylline 0 Oral
352 epinephrine 0 Subcutaneous
353 succinylcholine 0 Intravenous
354 thyrotropin alfa 0 Intramuscular
355 levorphanol 0 Oral
356 propantheline 0 Oral
357 carbinoxamine 0 Oral
358 diatrizoate 0 Intravenous
359 phytonadione 0 Oral
360 mecamylamine 0 Oral
361 liothyronine 0 Oral
362 methsuximide 0 Oral
363 mepenzolate 0 Oral
364 meclizine 0 Oral
365 triprolidine 0 Oral
366 benzonatate 1 Oral
367 Sodium polystyrene sulfonate 0 Oral
368 dichlorphenamide 0 Oral
369 phentermine 1 Oral
370 diethylpropion 0 Oral
371 oxymorphone 0 Oral
372 dexbrompheniramine 0 Oral
373 biperiden 0 Oral
374 isosorbide dinitrate 0 Oral
375 mepivacaine 0 Subcutaneous
376 bendroflumethiazide 1 Oral
377 phendimetrazine 0 Oral
378 oxytocin 0 Intravenous
379 guanethidine 0 Oral
380 ethosuximide 0 Oral
381 benzphetamine 0 Oral
382 glycopyrrolate 0 Oral
383 metyrapone 0 Oral
384 metaxalone 1 Oral
385 oxandrolone 1 Oral
386 oxazepam 0 Oral
387 protriptyline 0 Oral
388 cosyntropin 0 Intravenous
389 flavoxate 0 Oral
390 ketamine 1 Intravenous
391 pancuronium 0 Intravenous
392 pentagastrin 0 Intravenous
393 dextroamphetamine 0 Oral
394 terbutaline 1 Oral
395 calcitonin salmon 0 Subcutaneous
396 pentetic acid 0 Intravenous
397 nitroprusside 0 Intravenous
398 colestipol 0 Oral
399 lactulose 0 Oral
400 somatropin recombinant 0 Subcutaneous
401 fluorescein 0 Intravenous
402 metyrosine 0 Oral
403 carboprost tromethamine 0 Intramuscular
404 calcitriol 0 Oral
405 morphine 0 Oral
406 nabilone 0 Oral
407 vecuronium 0 Intravenous
408 atracurium 0 Intravenous
409 hydromorphone 0 Oral
410 sufentanil 0 Intravenous
411 tranexamic acid 0 Oral
412 alfentanil 0 Intravenous
413 ethanolamine oleate 0 Intravenous
414 rubidium chloride rb-82 0 Intravenous
415 urofollitropin 0 Subcutaneous
416 teriparatide 0 Subcutaneous
417 gadopentetate dimeglumine 0 Intravenous
418 rimantadine 0 Oral
419 pegademase bovine 0 Intramuscular
420 fenoldopam 0 Intravenous
421 calcium acetate 0 Oral
422 mivacurium 0 Intravenous
423 gadoteridol 0 Intravenous
424 enoxaparin 1 Subcutaneous
425 perindopril 0 Oral
426 rocuronium 0 Intravenous
427 dalteparin sodium 1 Subcutaneous
428 ferumoxsil 0 Oral
429 ferumoxides 0 Intravenous
430 porfimer 0 Intravenous
431 ibutilide 0 Intravenous
432 cisatracurium besylate 0 Intravenous
433 oxycodone 0 Oral
434 alendronate 1 Oral
435 tamsulosin 1 Oral
436 dolasetron 0 Oral
437 remifentanil 1 Intravenous
438 sibutramine 1 Oral
439 tiagabine 0 Oral
440 ropinirole 1 Oral
441 pramipexole 0 Oral
442 miglitol 0 Oral
443 polyethylene glycol 3350 0 Oral
444 delavirdine 0 Oral
445 tiludronate 0 Oral
446 eptifibatide 0 Intravenous
447 eprosartan 0 Oral
448 repaglinide 1 Oral
449 irbesartan 1 Oral
450 naratriptan 0 Oral
451 zolmitriptan 0 Oral
452 tolterodine 0 Oral
453 nelfinavir 1 Oral
454 rivastigmine 1 Oral
455 ziprasidone 1 Oral
456 risedronate 0 Oral
457 candesartan 1 Oral
458 clopidogrel 1 Oral
459 rizatriptan 0 Oral
460 bivalirudin 0 Intravenous
461 azacitidine 0 Intravenous
462 fluorouracil 1 Intravenous
463 argatroban 0 Intravenous
464 sildenafil 1 Oral
465 acarbose 1 Oral
466 acebutolol 1 Oral
467 tirofiban 0 Intravenous
468 sevelamer 0 Oral
469 dofetilide 0 Oral
470 acetylcysteine 0 Oral
471 acitretin 1 Oral
472 gadoversetamide 0 Intravenous
473 adenosine 0 Intravenous
474 salbutamol 0 Oral
475 almotriptan 0 Oral
476 frovatriptan 0 Oral
477 oxcarbazepine 1 Oral
478 rifapentine 0 Oral
479 levetiracetam 1 Oral
480 alpidem 1 Oral
481 bexarotene 1 Oral
482 perflutren 0 Intravenous
483 amifostine 0 Intravenous
484 amikacin 0 Intravenous
485 alosetron 1 Oral
486 aminocaproic acid 0 Oral
487 levothyroxine 1 Oral
488 linezolid 1 Intravenous
489 colesevelam 0 Oral
490 gemifloxacin 1 Oral
491 desloratadine 1 Oral
492 galantamine 0 Oral
493 cefditoren 0 Oral
494 zoledronate 1 Intravenous
495 caspofungin 0 Intravenous
496 atovaquone 0 Oral
497 voriconazole 1 Oral
498 guaifenesin 0 Oral
499 olmesartan 0 Oral
500 alfuzosin 1 Oral
501 aztreonam 0 Intravenous
502 dutasteride 0 Oral
503 baclofen 1 Oral
504 benazepril 1 Oral
505 bendazac 1 Oral
506 benzarone 1 Oral
507 benziodarone 1 Oral
508 ertapenem 0 Intravenous
509 benztropine 0 Oral
510 fondaparinux sodium 1 Subcutaneous
511 miglustat 0 Oral
512 gadobenate dimeglumine 0 Intravenous
513 rifaximin 0 Oral
514 tadalafil 0 Oral
515 palonosetron 0 Intravenous
516 betaxolol 0 Oral
517 vardenafil 0 Oral
518 bisoprolol 0 Oral
519 bleomycin 0 Intravenous
520 atomoxetine 1 Oral
521 bosentan 1 Oral
522 acamprosate 1 Oral
523 aripiprazole 0 Oral
524 budesonide 0 Oral
525 bumetanide 0 Oral
526 buspirone 0 Oral
527 eplerenone 0 Oral
528 butorphanol 0 Intravenous
529 cabergoline 0 Oral
530 ezetimibe 1 Oral
531 pregabalin 1 Oral
532 adefovir 1 Oral
533 ibandronate 0 Oral
534 carbenicillin 1 Oral
535 carbidopa 0 Oral
536 eszopiclone 0 Oral
537 cefaclor 1 Oral
538 cefadroxil 1 Oral
539 enfuvirtide 0 Subcutaneous
540 cefazolin 1 Intravenous
541 cefepime 1 Intravenous
542 cefixime 0 Oral
543 cefoperazone 1 Intravenous
544 cefotaxime 1 Intravenous
545 cefoxitin 0 Intravenous
546 cefpodoxime 0 Oral
547 oxaliplatin 1 Intravenous
548 cefprozil 1 Oral
549 ceftibuten 0 Oral
550 nitazoxanide 0 Oral
551 ceftriaxone 1 Intravenous
552 cefuroxime 1 Oral
553 micafungin 1 Intravenous
554 darifenacin 0 Oral
555 cephalexin 1 Oral
556 cetirizine 1 Oral
557 solifenacin 0 Oral
558 ranolazine 0 Oral
559 chloramphenicol 0 Intravenous
560 chlordiazepoxide 1 Oral
561 atazanavir 1 Oral
562 daptomycin 1 Intravenous
563 chlormezanone 1 Oral
564 bortezomib 1 Intravenous
565 anidulafungin 0 Intravenous
566 rasagiline 0 Oral
567 chloroquine 1 Oral
568 chlorothiazide 1 Oral
569 cinacalcet 0 Oral
570 conivaptan 0 Intravenous
571 nebivolol 0 Oral
572 chlorthalidone 0 Oral
573 erlotinib 1 Oral
574 alvimopan 0 Oral
575 cidofovir 0 Intravenous
576 ramelteon 0 Oral
577 cimetidine 1 Oral
578 cinchophen 1 Oral
579 tipranavir 1 Oral
580 tigecycline 0 Intravenous
581 cladribine 0 Intravenous
582 clindamycin 1 Oral
583 clometacin 1 Oral
584 urokinase 0 Intravenous
585 clonidine 0 Oral
586 nelarabine 1 Intravenous
587 cloxacillin 1 Oral
588 lenalidomide 1 Oral
589 lubiprostone 0 Oral
590 sorafenib 1 Oral
591 varenicline 1 Oral
592 darunavir 1 Oral
593 aliskiren 1 Oral
594 dasatinib 1 Oral
595 cyclobenzaprine 1 Oral
596 cyclofenil 1 Oral
597 sitagliptin 1 Oral
598 paliperidone 0 Oral
599 posaconazole 0 Oral
600 cyproheptadine 1 Oral
601 temsirolimus 0 Intravenous
602 tetrahydrobiopterin 0 Oral
603 milnacipran 1 Oral
604 desipramine 0 Oral
605 dexlansoprazole 1 Oral
606 everolimus 0 Oral
607 codeine 0 Oral
608 colistimethate 0 Intravenous
609 benzylpenicilloyl polylysine 0 Subcutaneous
610 cephradine 0 Oral
611 ceftizoxime 0 Intravenous
612 didanosine 1 Oral
613 mycophenolate mofetil 1 Oral
614 cefdinir 1 Oral
615 polymyxin b sulfate 0 Intravenous
616 diltiazem 1 Oral
617 sterile water 0 Intravenous
618 disopyramide 1 Oral
619 asparaginase 1 Intravenous
620 botulinum toxin type a 0 Intramuscular
621 interferon alfa-2b 1 Intravenous
622 dobutamine 0 Intravenous
623 docetaxel 1 Intravenous
624 interferon alfa-2a, recombinant 1 Subcutaneous
625 doxazosin 0 Oral
626 doxepin 1 Oral
627 alteplase 0 Intravenous
628 epoetin alfa 0 Intravenous
629 droperidol 0 Intravenous
630 droxicam 1 Oral
631 sargramostim 0 Intravenous
632 pegaspargase 1 Intravenous
633 efavirenz 1 Oral
634 muromonab-cd3 0 Intravenous
635 interferon beta-1b 1 Subcutaneous
636 abciximab 0 Intravenous
637 interferon beta-1a 1 Intramuscular
638 esmolol 0 Intravenous
639 estazolam 0 Oral
640 interferon alfacon-1 1 Subcutaneous
641 oprelvekin 0 Subcutaneous
642 estramustine 1 Oral
643 ethambutol 1 Oral
644 basiliximab 0 Intravenous
645 ethionamide 1 Oral
646 palivizumab 0 Intramuscular
647 infliximab 1 Intravenous
648 reteplase 0 Intravenous
649 trastuzumab 1 Intravenous
650 etanercept 1 Subcutaneous
651 etidronic acid 0 Oral
652 botulinum toxin type b 0 Intramuscular
653 etomidate 0 Intravenous
654 exifone 1 Oral
655 tenecteplase 0 Intravenous
656 rasburicase 0 Intravenous
657 alemtuzumab 0 Intravenous
658 peginterferon alfa-2b 1 Subcutaneous
659 fexofenadine 0 Oral
660 fialuridine 1 Oral
661 fipexide 1 Oral
662 anakinra 1 Subcutaneous
663 darbepoetin alfa 1 Intravenous
664 flecainide 1 Oral
665 omalizumab 0 Subcutaneous
666 ibritumomab tiuxetan 0 Intravenous
667 pegfilgrastim 0 Subcutaneous
668 flucytosine 0 Oral
669 fludarabine 0 Oral
670 flumazenil 0 Intravenous
671 adalimumab 1 Subcutaneous
672 cetuximab 0 Intravenous
673 bevacizumab 0 Intravenous
674 palifermin 0 Intravenous
675 natalizumab 1 Intravenous
676 flurazepam 1 Oral
677 fluvoxamine 0 Oral
678 foscarnet 0 Intravenous
679 fosfomycin 1 Oral
680 fosinopril 1 Oral
681 fosphenytoin 1 Intramuscular
682 galsulfase 0 Intravenous
683 abatacept 1 Intravenous
684 alglucosidase alfa 0 Intravenous
685 gemcitabine 1 Intravenous
686 panitumumab 0 Intravenous
687 idursulfase 0 Intravenous
688 certolizumab pegol 0 Subcutaneous
689 eculizumab 0 Intravenous
690 rilonacept 0 Subcutaneous
691 ustekinumab 0 Subcutaneous
692 romiplostim 0 Subcutaneous
693 ofatumumab 0 Intravenous
694 hydrochlorothiazide 1 Oral
695 idarubicin 0 Intravenous
696 indapamide 0 Oral
697 indinavir 0 Oral
698 iodipamide meglumine 0 Intravenous
699 irinotecan 1 Intravenous
700 l-methionine 0 Oral
701 isradipine 1 Oral
702 kanamycin 0 Intravenous
703 riboflavin 0 Oral
704 lamotrigine 1 Oral
705 l-carnitine 0 Oral
706 levofloxacin 1 Oral
707 levonorgestrel 0 Oral
708 lisinopril 1 Oral
709 loracarbef 1 Oral
710 loratadine 0 Oral
711 losartan 1 Oral
712 loxapine 0 Oral
713 mebanazine 1 Oral
714 mechlorethamine 0 Intravenous
715 mefloquine 1 Oral
716 vitamin e 0 Oral
717 melphalan 1 Oral
718 meprobamate 0 Oral
719 meropenem 1 Intravenous
720 methazolamide 1 Oral
721 methoxsalen 1 Oral
722 methylphenidate 1 Oral
723 methylscopolamine bromide 0 Oral
724 metoclopramide 1 Oral
725 mexiletine 1 Oral
726 midazolam 0 Oral
727 midodrine 0 Oral
728 mirtazapine 1 Oral
729 mitotane 0 Oral
730 mitoxantrone 1 Intravenous
731 moexipril 0 Oral
732 moxisylyte 1 Oral
733 folic acid 0 Oral
734 nabumetone 0 Oral
735 nadolol 0 Oral
736 nafcillin 1 Intravenous
737 nalbuphine 0 Intravenous
738 nialamide 1 Oral
739 nicardipine 0 Oral
740 nimodipine 0 Oral
741 niperotidine 1 Oral
742 nitroglycerin 0 Oral
743 nomifensine 1 Oral
744 norfloxacin 1 Oral
745 nortriptyline 1 Oral
746 octreotide 1 Intravenous
747 ondansetron 1 Oral
748 ofloxacin 1 Oral
749 diphenoxylate 0 Oral
750 oxacillin 1 Intravenous
751 ambenonium 0 Oral
752 papaverine 1 Intravenous
753 penbutolol 0 Oral
754 penicillin g 1 Intravenous
755 penicillin v 0 Oral
756 pentazocine 0 Intravenous
757 pentostatin 1 Intravenous
758 perphenazine 1 Oral
759 phenelzine 1 Oral
760 ephedrine 0 Intravenous
761 pimozide 0 Oral
762 pindolol 0 Oral
763 piperacillin 0 Intravenous
764 piroxicam 1 Oral
765 pirprofen 1 Oral
766 salsalate 1 Oral
767 polythiazide 0 Oral
768 probenecid 0 Oral
769 procainamide 1 Intravenous
770 propafenone 1 Oral
771 propranolol 0 Oral
772 propofol 1 Intravenous
773 pyrantel 0 Oral
774 pyrimethamine 1 Oral
775 quazepam 0 Oral
776 quinapril 1 Oral
777 quinidine 1 Oral
778 ramipril 1 Oral
779 reserpine 0 Oral
780 ribavirin 0 Oral
781 riluzole 1 Oral
782 risperidone 1 Oral
783 ritonavir 1 Oral
784 saquinavir 1 Oral
785 selegiline 0 Oral
786 succimer 1 Oral
787 sumatriptan 0 Oral
788 temazepam 0 Oral
789 teniposide 1 Intravenous
790 terazosin 0 Oral
791 thiotepa 1 Intravenous
792 timolol 0 Oral
793 sulcotidil 1 Oral
794 tolmetin 1 Oral
795 tolrestat 1 Oral
796 topotecan 0 Oral
797 tramadol 0 Oral
798 trandolapril 1 Oral
799 tranylcypromine 1 Oral
800 trazodone 1 Oral
801 triamterene 1 Oral
802 triazolam 0 Oral
803 trihexyphenidyl 0 Oral
804 trimethobenzamide 0 Oral
805 trimethoprim 1 Oral
806 fenclozic acid 1 Oral
807 ebrotidine 1 Oral
808 aceclofenac 1 Oral
809 nitrefazole 1 Oral
810 valaciclovir 1 Oral
811 valsartan 1 Oral
812 tetrabamate 1 Oral
813 vincristine 1 Intravenous
814 xenazoic acid 1 Oral
815 zafirlukast 1 Oral
816 falnidamol  1 Oral
817 zimelidine 1 Oral
818 caffeine 0 Intravenous
819 capreomycin 0 Intravenous
820 lidocaine 0 Oral
821 memantine 1 Oral
822 pamidronate 0 Intravenous
823 quinine 1 Oral
824 rosuvastatin 1 Oral
825 sulfamethizole 1 Oral
826 telithromycin 1 Oral
827 entacapone 1 Oral
828 valdecoxib 1 Oral
829 dexpanthenol 0 Intravenous
830 scopolamine 0 Intravenous
831 pyridoxine 0 Intravenous
832 thiamine 0 Intravenous
833 cyanocobalamin 0 Subcutaneous
834 cromoglicate 1 Oral
835 montelukast 1 Oral
836 moxifloxacin 1 Oral
837 vitamin c 0 Intravenous
838 sorbitol 0 Oral
839 capecitabine 0 Oral
840 leuprolide 1 Subcutaneous
841 eletriptan 0 Oral
842 hydroxychloroquine 1 Oral
843 ximelagatran 1 Oral
844 duloxetine 1 Oral
845 carisoprodol 0 Oral
846 dicloxacillin 1 Oral
847 metolazone 0 Oral
848 pamabrom 0 Oral
849 dextromethorphan 0 Oral
850 bacitracin 0 Intramuscular
851 paromomycin 0 Oral
852 telmisartan 1 Oral
853 ammonium chloride 0 Intravenous
854 amiloride 1 Oral
855 methysergide 0 Oral
856 methylergonovine 0 Oral
857 brompheniramine 0 Oral
858 l-arginine 0 Intravenous
859 pyridostigmine 0 Oral
860 phenoxybenzamine 0 Oral
861 oxybutynin 0 Oral
862 orphenadrine 0 Oral
863 loperamide 0 Oral
864 isoxsuprine 0 Oral
865 glafenine 1 Oral
866 acetylcholine chloride 0 Oral
867 amphetamine 1 Oral
868 mepazine 1 Oral
869 nandrolone decanoate 1 Intramuscular
870 auranofin 1 Oral
871 simethicone 0 Oral
872 betaine 0 Oral
873 bisacodyl 0 Oral
874 leucovorin 0 Oral
875 lapatinib 1 Oral
876 oseltamivir 0 Oral
877 alaproclate 1 Oral
878 orlistat 1 Oral
879 apomorphine 0 Subcutaneous
880 dihydroergotamine 0 Intravenous
881 procyclidine 0 Oral
882 clemastine 0 Oral
883 tenofovir 1 Oral
884 norethindrone acetate 0 Oral
885 exametazime 0 Intravenous
886 erythropoietin 0 Intravenous
887 Argipressin 0 Intravenous
888 sodium bicarbonate 0 Intravenous
889 plerixafor 0 Subcutaneous
890 tyramine 0 Oral
891 Hetastarch 0 Intravenous
892 imiglucerase 0 Intravenous
893 agalsidase beta 0 Intravenous
894 gadolinium ethoxybenzyl DTPA 0 Intravenous
895 canakinumab 1 Subcutaneous
896 Levoleucovorin 0 Intravenous
897 levomefolate calcium 0 Oral
898 sitaxsentan 1 Oral
899 dexmethylphenidate 1 Oral
900 hyaluronidase recombinant human 0 Subcutaneous
901 Androgenic steroids* 1  
902 Floxuridine 1 Intra-arterial
903 Flucloxacillin 1 oral
904 Halothane 1 Respiratory (inhalation)
905 Peginterferon 1  
906 Sulfonamides* 1 oral
907 Acetohexamide 1 oral
908 Dabigatran 1 oral
909 Gliclazide 1 Oral
910 Imipenem 1 Intravenous
911 Lopinavir 1 Oral
912 Molindone 1 Oral
913 Plicamycin 1  
914 Rilpivirine 1 Oral
915 Tibolone 1  
916 Tobramycin 1  
917 Vismodegib 1 Oral
918 Hydrocodone 0 Oral
919 Zalcitabine 0 Oral
920 Acrivastine 0 Oral
921 Amobarbital 0 Intramuscular; Intravenous, oral
922 Artemether 0 Oral
923 Bitolterol 0  
924 Butalbital 0 Oral
925 Butobarbital 0  
926 Carmustine 0 Intravenous
927 Chloral hydrate 0 Oral
928 Chlortetracycline 0 Tropical
929 Cilastatin 0 Intravenous
930 Cisapride 0 Oral
931 Cobicistat 0 Oral
932 Docusate 0 oral
933 Ergotamine 0 oral
934 Ethacrynate 0 oral
935 Fentanyl 0 Sublingual
936 Formoterol 0 Respiratory (inhalation)
937 Gentamicin 0 Intramuscular; Intravenous
938 Homatropine 0 Ophthalmic
939 Hyoscyamine 0 oral
940 Ipratropium 0 Oral; Respiratory (inhalation)
941 Levamisole 0 Oral
942 Levodopa 0 Oral
943 Liraglutide 0 Subcutaneous
944 Nalmefene 0 Oral
945 Pegaptanib 0 Intravitreal
946 Proguanil 0 Oral
947 Salmeterol 0 Oral; Respiratory (inhalation)
948 Tazobactam 0 Intravenous; Parenteral
949 Thiopental 0 Intravenous
950 Ticarcillin 0 Intramuscular; Intravenous
951 Tiotropium 0 Oral; Respiratory (inhalation)
952 Zanamivir 0 Oral; Respiratory (inhalation)
953 ACEMETACIN 1  
954 ACETARSOL 1 Vaginal
955 Alatrofloxacin 1  
956 Alimemazine 1 Oral
957 ANDROSTANOLONE 1  
958 Antithymocyte Immunoglobulin 1  
959 Artemisinin 1  
960 Artesunate 1  
961 bendazolic acid 1  
962 Bupivacaine 1 Epidural; Infiltration; Intracaudal; Perineural
963 CALCIUM CARBIMIDE 1 Oral
964 CARBIMAZOLE 1  
965 Cerivastatin 1 Oral
966 CILAZAPRIL 1 Oral
967 CINITAPRIDE 1  
968 Clomacron 1  
969 CLOMETHIAZOLE 1  
970 CLOTIAZEPAM 1  
971 COCAINE 1 Nasal, Torpical
972 CYPROTERONE 1 Oral, Intramuscular
973 Dehydroepiandrosterone 1  
974 Desflurane 1 Respiratory (inhalation)
975 DEXKETOPROFEN 1  
976 Diacetoxydiphenolisatin 1  
977 DICOUMAROL 1  
978 EBASTINE 1  
979 ENFLURANE 1 Respiratory (inhalation)
980 ESTRIOL 1  
981 Ethinylestradiol 1 Oral, Transdermal
982 ETRETINATE 1  
983 FLUPENTIXOL 1 Oral, Intramuscular
984 Fusidic Acid 1 Oral, Topical, Intravenous, optahlmic
985 Gemtuzumab 1  
986 GLUCOSAMINE 1 Topical
987 Growth Hormone 1 Intravenous
988 Interferon Unspecified 1  
989 Interferon-Beta-1a 1  
990 interferon-Beta-1b 1  
991 Ioxaglate And Meglumine 1 Intravascular
992 Isaxonine phosphate 1 Oral,Intramuscular; Intravenous
993 JOSAMYCIN 1  
994 LEVOMEPROMAZINE 1 Oral,Intramuscular; Intravenous
995 Melperone 1  
996 METAMIZOLE 1  
997 Methoxyflurane 1  
998 Methylene Dioxymethamphetamine 1  
999 NIFLUMIC ACID 1  
1000 Oxyiminoalkanoic acid derivative 1  
1001 Peginterferon-Alfa-2a 1  
1002 PENICILLIN 1  
1003 Phenisatin 1  
1004 Pivmecillinam 1 Oral
1005 RITODRINE 1 Oral, Intravenous
1006 ROFECOXIB 1 Oral
1007 ROXITHROMYCIN 1  
1008 STANOZOLOL 1  
1009 STREPTOKINASE 1 Intracoronary; Intravenous
1010 Suloctidil 1  
1011 TACRINE 1  
1012 TENOXICAM 1 Oral
1013 TIRATRICOL 1  
1014 TRIPTORELIN 1 Subcutaneous, Intramuscular
1015 phenacetin 1  
1016 bithionol 1  
1017 hexachlorophene 1 Topical
1018 methapyrilene 1  
1019 tripelennamine 1 Topical, Oral, vaginal
1020 oxyquinoline 1 oral, Topical,Vaginal, Dental
1021 meticillin 1  
1022 amsacrine 1 Intravenous
1023 furazolidone 1  
1024 hycanthone 1  
1025 idoxuridine 1 Opthalmic, Topical
1026 novobiocin 1  
1027 tianeptine 1  
1028 methacycline 1  
1029 bepridil 1  
1030 betahistine 1 Oral
1031 ciprofibrate 1  
1032 diethylcarbamazine 1 Oral
1033 fenoterol 1 Oral; Respiratory (inhalation)
1034 phenylbutazone 1 Oral
1035 ethynodiol diacetate 1 Oral
1036 atractyloside 1  
1037 temafloxacin 1  
1038 cefamandole 1 Intramuscular; Intravenous
1039 amodiaquine 1  
1040 glutethimide 1  
1041 sulfanilamide 1 Vaginal
1042 2-acetylaminofluorene 1  
1043 demecarium bromide 1  
1044 cefalotin 1 Intramuscular; Intravenous
1045 uracil mustard 1  
1046 methylphenobarbital 1  
1047 acenocoumarol 1 Oral
1048 1-naphthylisothiocyanate 1  
1049 aflatoxin b1 1  
1050 indacrinone 1  
1051 cefotiam 1  
1052 troleandomycin 1  
1053 perhexiline maleate 1  
1054 ciglitazone 1  
1055 fluspirilene 1 Intramuscular
1056 norgestrel 1 Oral
1057 carbon tetrachloride 1  
1058 aurothioglucose 1 Intramuscular
1059 phenothiazine 1  
1060 allyl alcohol 1  
1061 bromobenzene 1  
1062 azatadine 1 Oral
1063 allyl formate 1  
1064 tauroursodeoxycholic acid 1  
1065 octylmethoxycinnamate 1  
1066 ketotifen 0 Opthalmic, Topical
1067 permethrin 0 Topical
1068 oxyphenonium 0  
1069 pyridoxal phosphate 0 Oral
1070 aminoglutethimide 0 Oral
1071 tetracaine 0 Topical
1072 miconazole 0 Topical
1073 lindane 0 Topical
1074 astemizole 0 Oral
1075 ciclopirox 0 Topical
1076 pinacidil 0  
1077 terfenadine 0 Oral
1078 methoxamine 0 Intramuscular; Intravenous
1079 beclomethasone 0 Topical,Respiratory (inhalation)
1080 vidarabine 0  
1081 bezafibrate 0 oral
1082 bambuterol 0  
1083 gallamine triethiodide 0 Intravenous
1084 melatonin 0 Oral
1085 nocodazole 0  
1086 zomepirac 0  
1087 alloxan 0  
1088 pargyline 0  
1089 probucol 0 Oral
1090 lactose 0 Oral
1091 anileridine 0 Oral, Intramuscular; Intravenous; Subcutaneous
1092 citicoline 0  
1093 mometasone 0 Topical,Respiratory (inhalation)
1094 capsaicin 0 Percutaneous; Topical; Transdermal
1095 ergonovine 0 Oral, Intramuscular; Intravenous
1096 econazole 0 Topical
1097 sulconazole nitrate 0 Topical
1098 sulfabenzamide 0  
1099 cephapirin 0  
1100 azlocillin 0  
1101 butoconazole 0 Vaginal
1102 mibefradil 0  
1103 ragaglitazar 0  
1104 bismuth subsalicylate 0 Oral
1105 isoxicam 0  
1106 inositol 0 Oral, Vaginal
1107 latamoxef 0  
1108 Abiraterone 1  
1109 Acetorphan 1  
1110 Alfacalcidol 1  
1111 Ambroxol 1  
1112 Aminolevulinic acid 1  
1113 Amisulpride 1  
1114 Ampiroxicam 1  
1115 Anethole 1  
1116 Arbekacin 1  
1117 Axitinib 1  
1118 Azelnidipine 1  
1119 Bacampicillin 1  
1120 Benidipine 1  
1121 Beraprost 1  
1122 Boceprevir 1  
1123 Bromazepam 1  
1124 Bromhexine 1  
1125 Bromisoval 1  
1126 Brotizolam 1  
1127 Bucillamine 1  
1128 Buflomedil 1  
1129 Buprenorphine 1  
1130 Cabazitaxel 1  
1131 Cefcapene 1  
1132 Cefmetazole 1  
1133 Cefozopran 1  
1134 Cefpirome 1  
1135 Celiprolol 1  
1136 Chlormadinone 1  
1137 Cibenzoline 1  
1138 Cilnidipine 1  
1139 Clobazam 1  
1140 Clobetasol 1  
1141 Clodronic acid 1  
1142 Clofazimine 1  
1143 Cloperastine 1  
1144 Crizotinib 1  
1145 Curcumin 1  
1146 Cyamemazine 1  
1147 Cyclothiazide 1  
1148 Desogestrel 1  
1149 Diacerein 1  
1150 Dihydrocodeine 1  
1151 Dirithromycin 1  
1152 Domperidone 1  
1153 Doxifluridine 1  
1154 Droxidopa 1  
1155 Dydrogesterone 1  
1156 Edaravone 1  
1157 Eltrombopag 1  
1158 Eperisone 1  
1159 Epinastine 1  
1160 Eribulin Mesylate 1  
1161 Ethanol 1  
1162 Ethyl loflazepate 1  
1163 Ethylene glycol 1  
1164 Etizolam 1  
1165 Etoricoxib 1  
1166 Flomoxef 1  
1167 Fluindione 1  
1168 Flunitrazepam 1  
1169 Flupirtine 1  
1170 Fominoben 1  
1171 Fosfluconazole 1  
1172 Fudosteine 1  
1173 Gabapentin Enacarbil 1  
1174 Gabexate 1  
1175 Garenoxacin 1  
1176 Glutathione 1  
1177 Glycerol 1  
1178 Glycyrrhizin 1  
1179 Halofantrine 1  
1180 Heptaminol 1  
1181 Hypericin 1  
1182 Ibudilast 1  
1183 Iloprost 1  
1184 Irsogladine 1  
1185 Isepamicin 1  
1186 Isosorbide 1  
1187 Itopride 1  
1188 Lafutidine 1  
1189 Lanreotide 1  
1190 Lercanidipine 1  
1191 Levocetirizine 1  
1192 Lodenosine 1  
1193 Lormetazepam 1  
1194 Lornoxicam 1  
1195 Loxoprofen 1  
1196 Manidipine 1  
1197 Mazindol 1  
1198 Menatetrenone 1  
1199 Mequitazine 1  
1200 Metopimazine 1  
1201 Mitiglinide 1  
1202 Mizoribine 1  
1203 Molsidomine 1  
1204 Mosapride 1  
1205 Moxonidine 1  
1206 Nafamostat 1  
1207 Naftidrofuryl 1  
1208 Nandrolone 1  
1209 Nefopam 1  
1210 Netilmicin 1  
1211 Nicergoline 1  
1212 Nicorandil 1  
1213 Nitrazepam 1  
1214 Nitrendipine 1  
1215 Nordazepam 1  
1216 Norethisterone 1  
1217 Olopatadine 1  
1218 Oxatomide 1  
1219 Oxyphenbutazone 1  
1220 Ozagrel 1  
1221 Pazufloxacin 1  
1222 Peramivir 1  
1223 Phenformin 1  
1224 Phenprocoumon 1  
1225 Phenylephrine 1  
1226 Phloroglucinol 1  
1227 Picolamine 1  
1228 Pilsicainide 1  
1229 Pimecrolimus 1  
1230 Pinaverium 1  
1231 Piperacetazine 1  
1232 Pipobroman 1  
1233 Piracetam 1  
1234 Pirarubicin 1  
1235 Pranlukast 1  
1236 Pranoprofen 1  
1237 Prazepam 1  
1238 Propacetamol 1  
1239 Propiverine 1  
1240 Raltitrexed 1  
1241 Rebamipide 1  
1242 Rilmenidine 1  
1243 Rivaroxaban 1  
1244 Roxatidine 1  
1245 Salicylic acid 1  
1246 Sarpogrelate 1  
1247 Sennoside 1  
1248 Sofalcone 1  
1249 Sparfloxacin 1  
1250 Sulfamethoxazole 1  
1251 Sulpiride 1  
1252 Suplatast 1  
1253 Tandospirone 1  
1254 Telaprevir 1  
1255 Temocapril 1  
1256 Teprenone 1  
1257 Tetrazepam 1  
1258 Theobromine 1  
1259 Thiocolchicoside 1  
1260 Tiapride 1  
1261 Tiaprofenic acid 1  
1262 Tiquizium 1  
1263 Tocainide 1  
1264 Trabectedin 1  
1265 Tranilast 1  
1266 Trapidil 1  
1267 Trichlormethiazide 1  
1268 Trimebutine 1  
1269 Trimetazidine 1  
1270 Tropatepine 1  
1271 Troxipide 1  
1272 Urapidil 1  
1273 Valpromide 1  
1274 Vemurafenib 1  
1275 Vindesine 1  
1276 Voglibose 1  
1277 Xylometazoline 1  
1278 Zaltoprofen 1  
1279 Zopiclone 1  

 

 

 

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